SCHEMBL6587557

SCHEMBL6587557

Cc1cc(-c2ccc(NC(=O)NC3CC3C3CCCCC3)c3ccccc23)cc(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
KMT2A Q03164 2/20 0.36
CHRM2 P08172 2/20 0.36
CHRM1 P11229 2/20 0.36
CHRM3 P20309 2/20 0.36
SHMT2 P34897 2/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
TAS1R3 Q7RTX0 2/20 0.35
TAS1R1 Q7RTX1 2/20 0.35
EPHX2 P34913 1/20 0.34
PARP1 P09874 1/20 0.34
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
CXCR2 P25025 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6588782 0.80 EPHX1 (0.38) EPHX1TRPV1KMT2ACHRM2CHRM1
SCHEMBL5752633 0.73 PI4KA (0.39) EPHX1CHRM2CHRM1CHRM3SHMT2
SCHEMBL6583944 0.71 KDR (0.40) EPHX1TRPV1
SCHEMBL6810815 0.71 KDR (0.42) EPHX1KMT2ASMN1; SMN2TAS1R3TAS1R1
SCHEMBL5753008 0.70 MAPK14 (0.56) CHRM2CHRM1CHRM3
SCHEMBL6583491 0.70 KDR (0.39) EPHX1KMT2AHTTSMN1; SMN2MEN1
SCHEMBL6589214 0.70 KDR (0.41) EPHX1KMT2ATAS1R3TAS1R1
SCHEMBL6586069 0.69 EPHX1 (0.39) EPHX1TRPV1KMT2ASHMT2HTT
SCHEMBL6598212 0.69 KDR (0.40) EPHX1
SCHEMBL6583664 0.69 KDR (0.40) EPHX1KMT2ASHMT2SMN1; SMN2TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004534787-A 2004-11-18 JP claimed
EP-1414810-A2 1,4-DISUBSTITUTED BENZO-FUSED CYCLOALKYL UREA COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-05-06 EP claimed
WO-2002098869-A2 1,4-DISUBSTITUTED BENZO-FUSED CYCLOALKYL UREA COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-12 WO claimed