SCHEMBL6587679

SCHEMBL6587679

NC(=O)Oc1cccc2[nH]c(-c3ccc(N4CCOCC4)nc3)nc12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.53
AURKB Q96GD4 2/20 0.53
KDR P35968 1/20 0.53
ATR Q13535 2/20 0.49
DGAT1 O75907 3/20 0.48
KCNH2 Q12809 3/20 0.48
ADORA2A P29274 1/20 0.48
PARP1 P09874 6/20 0.47
JAK2 O60674 1/20 0.47
SOAT1 P35610 1/20 0.45
CNR2 P34972 5/20 0.43
DHODH Q02127 1/20 0.43
TDO2 P48775 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587264 0.91 AURKA (0.55) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587512 0.90 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587278 0.90 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6586056 0.90 AURKA (0.59) AURKAAURKBKDRATRDGAT1
SCHEMBL6588365 0.89 AURKA (0.54) AURKAAURKBKDRATRDGAT1
SCHEMBL6590217 0.89 AURKA (0.59) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6589042 0.87 AURKA (0.56) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587702 0.86 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6591285 0.86 AURKA (0.51) AURKAAURKBKDRATRDGAT1
SCHEMBL6588603 0.86 AURKA (0.63) AURKAAURKBKDRDGAT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed