SCHEMBL6592073

SCHEMBL6592073

COC(=O)c1cccc(-c2ccc(C=Cc3cc(C(F)(F)F)[nH]c(=O)n3)o2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.62
MEN1 O00255 5/20 0.62
POLB P06746 5/20 0.62
MAPT P10636 4/20 0.62
LMNA P02545 3/20 0.62
HPGD P15428 2/20 0.62
PSD A5PKW4 1/20 0.61
ALDH1A1 P00352 8/20 0.59
KDM4E B2RXH2 7/20 0.59
USP2 O75604 2/20 0.59
HTT P42858 1/20 0.59
RECQL P46063 1/20 0.59
TLR9 Q9NR96 1/20 0.59
CRHBP P24387 1/20 0.55
CRHR2 Q13324 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
PIK3CG P48736 1/20 0.49
XPA P23025 1/20 0.49
TNF P01375 2/20 0.44
NOD1 Q9Y239 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6592069 1.00 KMT2A (0.62) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6593873 0.89 POLB (0.68) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6593877 0.89 POLB (0.68) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6593648 0.82 PSD (0.82) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6593640 0.82 PSD (0.82) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6597395 0.80 MEN1 (0.77) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6597397 0.80 MEN1 (0.77) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6595066 0.79 MAPT (0.66) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6595069 0.79 MAPT (0.66) KMT2AMEN1POLBMAPTLMNA
SCHEMBL6593705 0.78 PSD (0.69) KMT2AMEN1POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004016271-A1 PYRIMIDONES AS ANTIVIRAL AGENTS AXXIMA PHARMACEUTICALS AG (DE) 2004-02-26 WO claimed
EP-1389461-A1 Pyrimidones with antiviral properties Axxima Pharmaceuticals Aktiengesellschaft (DE) 2004-02-18 EP claimed
WO-2004016271-A1 PYRIMIDONES AS ANTIVIRAL AGENTS AXXIMA PHARMACEUTICALS AG (DE) 2004-02-26 WO disclosed
EP-1389461-A1 Pyrimidones with antiviral properties Axxima Pharmaceuticals Aktiengesellschaft (DE) 2004-02-18 EP disclosed