SCHEMBL6594022

SCHEMBL6594022

CCCCCn1c(N2CCCN(CCC(CN(C)C(=O)c3ccc(OC)cc3OC)c3ccc(Cl)c(Cl)c3)CC2)nc2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 13/20 0.47
TACR1 P25103 1/20 0.45
TACR3 P29371 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6593919 0.93 TACR2 (0.47) TACR2TACR1TACR3
SCHEMBL6599260 0.89 TACR2 (0.52) TACR2TACR1
SCHEMBL6599776 0.89 TACR2 (0.45) TACR2TACR1TACR3
SCHEMBL6599086 0.89 TACR2 (0.45) TACR2TACR1TACR3
SCHEMBL6599098 0.88 TACR2 (0.45) TACR2TACR1TACR3
SCHEMBL6598484 0.88 TACR2 (0.45) TACR2TACR1TACR3
SCHEMBL6597245 0.87 TACR2 (0.64) TACR2TACR1
SCHEMBL6597363 0.86 TACR2 (0.58) TACR2TACR1
SCHEMBL6596914 0.86 TACR2 (0.44) TACR2
SCHEMBL6596639 0.86 TACR2 (0.43) TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888338-B1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL) 1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES AVENTIS PHARMA INC (US) 2004-11-17 EP disclosed