Benzene

Benzene

SCHEMBL6594689

C#Cc1c(C(=O)O)nc2c(OC)cccc2c1O.c1ccccc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.46
CDK9 P50750 1/20 0.42
DYRK1A Q13627 1/20 0.42
TNKS O95271 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
KDM4E B2RXH2 4/20 0.38
ADORA2A P29274 5/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
HSD17B10 Q99714 1/20 0.38
ALOX15 P16050 1/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080920 0.81 PDE10A (0.50) PDE10ACDK9DYRK1ATNKSTNKS2
SCHEMBL6080957 0.75 PDE10A (0.52) PDE10ACDK9DYRK1ATNKSTNKS2
SCHEMBL6080303 0.73 KDM5B (0.36) ADORA2A
SCHEMBL6081023 0.72 KDM4E (0.52) PDE10ACDK9DYRK1ATNKSTNKS2
SCHEMBL27276202 0.72 CA12 (0.50) PDE10ACDK9DYRK1ATNKSTNKS2
SCHEMBL6594661 0.72 DUSP3 (0.41) KDM4EALDH1A1ALOX15MEN1GAA
SCHEMBL17966023 0.71 ADORA2A (0.61) ADORA2A
SCHEMBL24010068 0.70 KDM4E (0.47) KDM4EALDH1A1HPGDHSD17B10THRB
SCHEMBL2924449 0.70 NQO2 (0.59) PDE10ATNKSTNKS2PARP2ALDH1A1
SCHEMBL6081016 0.70 PDE10A (0.56) PDE10ACDK9DYRK1ATNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed