SCHEMBL6594944

SCHEMBL6594944

O=C(c1ccc(OCCN2CCCC2)cc1)c1c(-c2ccc(CCCN3CCCC3)cc2)sc2ccccc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.79
ESR2 Q92731 16/20 0.79
F2 P00734 1/20 0.72
HDAC1 Q13547 3/20 0.66
HDAC6 Q9UBN7 3/20 0.66
MEN1 O00255 1/20 0.66
PLD2 O14939 1/20 0.66
KDM1A O60341 1/20 0.66
NR1I2 O75469 1/20 0.66
USP2 O75604 1/20 0.66
ALDH1A1 P00352 1/20 0.66
C5 P01031 1/20 0.66
LMNA P02545 1/20 0.66
TP53 P04637 1/20 0.66
FYN P06241 1/20 0.66
PGR P06401 1/20 0.66
CYP3A4 P08684 1/20 0.66
ADRA2A P08913 1/20 0.66
ADORA3 P0DMS8 1/20 0.66
CYP2D6 P10635 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595171 1.00 ESR1 (0.79) ESR1ESR2F2HDAC1HDAC6
SCHEMBL7772287 0.94 ESR1 (0.82) ESR1ESR2F2HDAC1HDAC6
SCHEMBL7451884 0.93 ESR1 (0.87) ESR1ESR2F2MEN1PLD2
SCHEMBL7775840 0.93 ESR1 (0.87) ESR1ESR2F2MEN1PLD2
SCHEMBL7774124 0.93 ESR1 (0.85) ESR1ESR2F2MEN1PLD2
SCHEMBL6595547 0.92 ESR1 (0.92) ESR1ESR2F2MEN1PLD2
SCHEMBL6597972 0.92 ESR1 (0.94) ESR1ESR2F2MEN1PLD2
SCHEMBL6595743 0.92 ESR1 (0.94) ESR1ESR2F2MEN1PLD2
SCHEMBL6591897 0.91 ESR1 (0.82) ESR1ESR2F2MEN1PLD2
SCHEMBL6595868 0.90 ESR1 (0.83) ESR1ESR2F2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed