SCHEMBL6596500

SCHEMBL6596500

Cc1nc(C)n(C)c1-c1ccnc(Nc2ccccc2)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 8/20 0.64
CDK4 P11802 4/20 0.64
CCNE1 P24864 1/20 0.64
KDR P35968 8/20 0.63
PTK2 Q05397 7/20 0.63
PLK1 P53350 4/20 0.63
AURKB Q96GD4 3/20 0.52
AKT1 P31749 2/20 0.52
PRKCD Q05655 2/20 0.50
ABL1 P00519 1/20 0.50
EGFR P00533 1/20 0.50
PRKCA P17252 1/20 0.50
CHEK1 O14757 1/20 0.48
IKBKB O14920 1/20 0.48
AURKA O14965 1/20 0.48
NPC1 O15118 1/20 0.48
PDPK1 O15530 1/20 0.48
CHEK2 O96017 1/20 0.48
PRKCG P05129 1/20 0.48
CDK1 P06493 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4819158 0.83 CDK2 (0.60) CDK2CDK4CCNE1KDRPTK2
SCHEMBL6593928 0.82 CDK2 (0.69) CDK2CDK4IKBKBCDK1JAK2
SCHEMBL6596039 0.81 CDK2 (0.72) CDK2CDK4CCNE1KDRPTK2
SCHEMBL5105343 0.78 CDK2 (0.69) CDK2CDK4CCNE1KDRPTK2
SCHEMBL6593019 0.78 CDK2 (0.68) CDK2CDK4CCNE1KDRPTK2
SCHEMBL6245628 0.77 CDK2 (0.69) CDK2CDK4CCNE1KDRPTK2
SCHEMBL6598042 0.77 CDK2 (0.66) CDK2CDK4CCNE1PLK1IKBKB
SCHEMBL4826063 0.76 CDK2 (0.58) CDK2CDK4CCNE1KDRPTK2
Dimethylamine SCHEMBL6593494 0.75 CDK2 (0.78) CDK2CDK4IKBKBCDK1
SCHEMBL1593016 0.73 PRKCD (0.79) CDK2CDK4PLK1PRKCDABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1269813-C Imidazolo-5-yl-2-anilino-pyrimidines as agents for inhibition of cell proliferation ASTRAZENECA AB (SE) 2006-08-16 CN disclosed
EP-1351958-B1 IMIDAZOLO-5-YL-2-ANILINO-PYRIMIDINES AS AGENTS FOR THE INHIBITION OF THE CELL PROLIFERATION ASTRAZENECA AB (SE) 2004-06-16 EP disclosed