SCHEMBL6596548

SCHEMBL6596548

COc1cc(C(=O)N(C)CC(CCN2CCCN(c3nc4ccccc4n3Cc3cccs3)CC2)c2ccccc2)cc(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 1/20 0.42
TACR2 P21452 4/20 0.40
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
TACR1 P25103 1/20 0.37
PYGM P11217 1/20 0.37
SLC29A1 Q99808 1/20 0.37
ABCC1 P33527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6596687 0.89 TACR2 (0.43) ALDH1A1LMNATACR2MAPTTACR1
SCHEMBL6594153 0.89 HRH1 (0.45) ALDH1A1LMNAHTTTACR2MAPT
SCHEMBL6597168 0.88 TACR2 (0.39) ALDH1A1LMNATACR2MAPTTSHR
SCHEMBL6599725 0.88 TACR2 (0.39) ALDH1A1LMNATACR2MAPTTACR1
SCHEMBL6599093 0.88 TACR2 (0.46) TACR2TSHRTACR1SLC29A1
SCHEMBL8448809 0.88 TACR2 (0.40) ALDH1A1LMNAHTTTACR2MAPT
SCHEMBL6594042 0.88 HRH1 (0.44) TACR2TACR1SLC29A1
SCHEMBL6596465 0.88 HRH1 (0.45) TACR2TACR1
SCHEMBL6596448 0.87 TACR2 (0.41) ALDH1A1LMNATACR2MAPT
SCHEMBL6596863 0.87 TACR2 (0.41) ALDH1A1LMNATACR2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888338-B1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL) 1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES AVENTIS PHARMA INC (US) 2004-11-17 EP disclosed
EP-0612750-B1 Cephalosporinderivatives BIOCHEMIE GMBH (AT) 1999-03-03 EP disclosed
EP-0888338-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL) 1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1999-01-07 EP disclosed
WO-1997030991-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL)[1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1997-08-28 WO disclosed
EP-0612750-A2 Cephalosporinderivatives BIOCHEMIE Gesellschaft m.b.H. (AT) 1994-08-31 EP disclosed
EP-0204781-A1 NEW PROCESS FOR PROCUDING CEPHALOSPORINE DERIVATIVES. BIOCHEMIE GMBH (AT) 1986-12-17 EP disclosed
WO-1986003204-A1 NEW PROCESS FOR PROCUDING CEPHALOSPORINE DERIVATIVES BIOCHEMIE GESELLSCHAFT M.B.H. (AT) 1986-06-05 WO disclosed