SCHEMBL6597011

SCHEMBL6597011

Nc1ncc(-c2ccc(S(=O)(=O)NCCN3CCCC3)cc2)nc1C(=O)Nc1cccnc1

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.73
CCNE2 O96020 13/20 0.73
CCNE1 P24864 13/20 0.73
CDK2 P24941 13/20 0.73
GSK3A P49840 1/20 0.66
ATR Q13535 5/20 0.62
ATRIP Q8WXE1 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6034611 0.99 GSK3B (0.72) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL6034231 0.95 GSK3B (0.71) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL6035843 0.88 GSK3B (0.71) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL6034766 0.88 GSK3B (0.71) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL6034644 0.86 ATR (0.84) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL6035259 0.85 GSK3B (0.66) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL6034152 0.85 ATR (0.84) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL3149256 0.85 ATR (0.82) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL31061310 0.85 GSK3B (1.00) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL31259907 0.85 GSK3B (1.00) GSK3BCCNE2CCNE1CDK2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP claimed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO claimed
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP disclosed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO disclosed