SCHEMBL6597791

SCHEMBL6597791

CN(CC(CCN1CCCN(c2nc3ccccc3n2Cc2ccoc2)CC1)c1ccc2c(c1)OCO2)C(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 14/20 0.46
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MCL1 Q07820 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CCR5 P51681 1/20 0.40
TACR1 P25103 1/20 0.40
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6599095 0.92 HRH1 (0.39) TACR2ALDH1A1KDM4EMCL1L3MBTL1
SCHEMBL6598098 0.91 TACR2 (0.48) TACR2TACR1
SCHEMBL6595957 0.91 TACR2 (0.46) TACR2TACR1
SCHEMBL6595836 0.90 TACR2 (0.59) TACR2TACR1
SCHEMBL6597483 0.90 TACR2 (0.47) TACR2TACR1
SCHEMBL6596135 0.89 TACR2 (0.46) TACR2ALDH1A1KDM4EMCL1L3MBTL1
SCHEMBL6598925 0.89 TACR2 (0.48) TACR2KDM4ETACR1MAPK1
SCHEMBL6599166 0.89 TACR2 (0.45) TACR2
SCHEMBL6593512 0.89 TACR2 (0.46) TACR2TACR1
SCHEMBL6599556 0.89 TACR2 (0.48) TACR2CCR5TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888338-B1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL) 1,4]DIAZEPAN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES AVENTIS PHARMA INC (US) 2004-11-17 EP disclosed