SCHEMBL6598538

SCHEMBL6598538

COc1cc2sc(-c3ccc(OCCN4CCCC4)cc3)c(C(=O)c3ccc(O[C@H]4CCCC[C@@H]4N4CCCCC4)cc3)c2cc1F

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.62
ESR2 Q92731 19/20 0.62
ENPP3 O14638 1/20 0.56
MEN1 O00255 2/20 0.56
ALDH1A1 P00352 2/20 0.56
LMNA P02545 2/20 0.56
TP53 P04637 2/20 0.56
CYP3A4 P08684 2/20 0.56
MAPT P10636 2/20 0.56
ALOX15 P16050 2/20 0.56
KMT2A Q03164 2/20 0.56
HSD17B10 Q99714 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
PLD2 O14939 1/20 0.56
KDM1A O60341 1/20 0.56
NR1I2 O75469 1/20 0.56
USP2 O75604 1/20 0.56
C5 P01031 1/20 0.56
FYN P06241 1/20 0.56
PGR P06401 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6598546 1.00 ESR1 (0.62) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6598543 1.00 ESR1 (0.62) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6594987 0.90 ESR1 (0.77) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6594981 0.90 ESR1 (0.77) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6594975 0.90 ESR1 (0.77) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6596695 0.89 ESR1 (0.73) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL6597301 0.89 ESR1 (0.79) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6597302 0.89 ESR1 (0.79) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6591884 0.89 ESR1 (0.79) ESR1ESR2ENPP3MEN1ALDH1A1
SCHEMBL6597305 0.89 ESR1 (0.79) ESR1ESR2ENPP3MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed