SCHEMBL6599253

SCHEMBL6599253

CC(C)(C)c1csc(-c2cc3cc(Cn4nc(C(N)=O)c5cc(OCc6ccccc6)ccc54)ccc3o2)n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 4/20 0.39
PLA2G2A P14555 1/20 0.37
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
FAAH O00519 2/20 0.34
MGLL Q99685 2/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
HIF1A Q16665 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN12 Q05209 1/20 0.34
PTPN22 Q9Y2R2 1/20 0.34
S1PR1 P21453 1/20 0.34
PKM P14618 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600128 0.90 F2RL3 (0.37) F2RL3PLA2G2ACASP3SENP8SENP7
SCHEMBL6597890 0.90 MAOB (0.40) F2RL3PLA2G2A
SCHEMBL7533433 0.87 APP (0.35)
SCHEMBL6599144 0.87 CPT1A (0.39)
SCHEMBL6601063 0.85 MCL1 (0.40) F2RL3S1PR1PKM
SCHEMBL7469206 0.84 MAOB (0.31)
SCHEMBL6603445 0.83 CPT1A (0.38) F2RL3
SCHEMBL6601472 0.82 KMT2A (0.40) F2RL3PLA2G2A
SCHEMBL5810419 0.82 PPARD (0.53) F2RL3PLA2G2A
SCHEMBL8659965 0.82 MEN1 (0.40) HIF1APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1170009-B1 Thiazolybenzofuran derivatives and their use as SRS-A and leukotiene antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2004-04-07 EP disclosed
EP-1170009-A2 Thiazolybenzofuran derivatives and their use as SRS-A and leukotiene antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-09 EP disclosed
US-5994378-A ANTIALLERGENS; ANTIINFLAMMATORY AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-11-30 US disclosed
EP-0880519-A1 THIAZOLYLBENZOFURAN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-12-02 EP disclosed
WO-1997027190-A1 THIAZOLYLBENZOFURAN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-31 WO disclosed