SCHEMBL6599358

SCHEMBL6599358

CN(C)CCN(C)C(=O)c1ccc(-c2cnc(N)c(C(=O)Nc3cccnc3)n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 1.00
CCNE2 O96020 8/20 1.00
CCNE1 P24864 8/20 1.00
CDK2 P24941 8/20 1.00
ATR Q13535 11/20 0.83
CYP3A4 P08684 1/20 0.58
GSK3A P49840 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6035742 0.99 GSK3B (0.98) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6034278 0.95 GSK3B (0.90) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6034146 0.91 GSK3B (0.84) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL2483383 0.91 ATR (1.00) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6034005 0.87 CCNE2 (0.77) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6034567 0.86 GSK3B (0.75) GSK3BCCNE2CCNE1CDK2ATR
Hydrochloric Acid SCHEMBL6597556 0.85 GSK3B (0.74) GSK3BCCNE2CCNE1CDK2ATR
Hydrochloric Acid SCHEMBL6033864 0.84 GSK3B (0.72) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL6616717 0.82 ATR (0.82) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL3162088 0.82 ATR (0.81) GSK3BCCNE2CCNE1CDK2ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP claimed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO claimed
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP disclosed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO disclosed