SCHEMBL6599474

SCHEMBL6599474

COc1cc(C(=O)c2c(-c3ccc(CCN4CCCC4)cc3)sc3cc(OCc4ccccc4)ccc23)ccc1CN1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.55
ESR2 Q92731 16/20 0.55
F2 P00734 3/20 0.53
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597513 0.96 ESR1 (0.59) ESR1ESR2F2HDAC1HDAC6
SCHEMBL6596715 0.93 ESR1 (0.60) ESR1ESR2F2
SCHEMBL7774110 0.92 ESR1 (0.48) ESR1ESR2F2
SCHEMBL6594992 0.90 ESR1 (0.55) ESR1ESR2F2
SCHEMBL6174247 0.89 F2 (0.57) ESR1ESR2F2
SCHEMBL6171544 0.89 F2 (0.53) ESR1ESR2F2
SCHEMBL6172249 0.89 ESR1 (0.50) ESR1ESR2F2
SCHEMBL6592408 0.89 ESR1 (0.65) ESR1ESR2F2
SCHEMBL6596359 0.89 F2 (0.67) ESR1ESR2F2HDAC1HDAC6
SCHEMBL7775991 0.89 ESR1 (0.55) ESR1ESR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed