SCHEMBL6602020

SCHEMBL6602020

COc1ccc(-c2sc3cc(OC)ccc3c2C(=O)c2ccc(OC3CCN(Cc4ccccc4)C3)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.56
ESR2 Q92731 13/20 0.56
CNR1 P21554 1/20 0.52
CNR2 P34972 1/20 0.52
CHEK2 O96017 1/20 0.49
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48
TUBB2A Q13885 1/20 0.48
TUBB8 Q3ZCM7 1/20 0.48
TUBA3E Q6PEY2 1/20 0.48
TUBA1A Q71U36 1/20 0.48
TUBA1C Q9BQE3 1/20 0.48
TUBB6 Q9BUF5 1/20 0.48
TUBB2B Q9BVA1 1/20 0.48
TUBB1 Q9H4B7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600990 0.95 ESR1 (0.58) ESR1ESR2CNR1CNR2CHEK2
SCHEMBL6601476 0.89 ESR1 (0.66) ESR1ESR2CNR1ACHE
SCHEMBL6602854 0.88 ESR1 (0.65) ESR1ESR2CNR1CNR2ENPP3
SCHEMBL6600800 0.85 ESR1 (0.61) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL6602789 0.84 ESR1 (0.62) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL6601827 0.84 ESR1 (0.70) ESR1ESR2CNR1ACHE
SCHEMBL6603461 0.84 ESR1 (0.63) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL8490502 0.82 CHEK2 (0.53) CHEK2BCHEACHE
SCHEMBL6601882 0.81 ESR1 (0.56) ESR1ESR2CNR1ACHE
SCHEMBL6601102 0.81 ESR1 (0.61) ESR1ESR2CNR1CNR2TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0905132-B1 Benzothiophenes LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6060488-A ANTICARCINOGENIC AGENTS; POSTMENOPAUSAL CANCER OF BREASTS, UTERUS, CERVIX ELI LILLY AND COMPANY (US) 2000-05-09 US disclosed
EP-0905132-A1 Benzothiophenes ELI LILLY AND COMPANY (US) 1999-03-31 EP disclosed