SCHEMBL6603510

SCHEMBL6603510

COc1ccc(NC(=O)c2ccc(-c3ccncc3)c(C)c2)cc1OCCN(C)C

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.69
HTR1B P28222 9/20 0.69
HTR2A P28223 5/20 0.69
MEN1 O00255 2/20 0.69
ALDH1A1 P00352 2/20 0.69
KMT2A Q03164 2/20 0.69
KDM4E B2RXH2 1/20 0.69
TP53 P04637 1/20 0.69
CYP1A2 P05177 1/20 0.69
CYP3A4 P08684 1/20 0.69
CYP2D6 P10635 1/20 0.69
MAPT P10636 1/20 0.69
HPGD P15428 1/20 0.69
ALOX15 P16050 1/20 0.69
MAPK1 P28482 1/20 0.69
HSD17B10 Q99714 1/20 0.69
TDP1 Q9NUW8 1/20 0.69
CHRM2 P08172 1/20 0.68
ADRA2A P08913 1/20 0.68
CHRM1 P11229 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744156 0.89 HTR1D (0.72) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8654316 0.89 HTR1D (0.74) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8653043 0.88 HTR1D (0.73) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL7447318 0.88 HTR1D (0.66) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL7397448 0.85 HTR1D (0.69) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL7450572 0.85 HTR1D (0.91) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8652789 0.85 HTR1D (0.69) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8662120 0.85 HTR1D (0.69) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8652792 0.85 HTR1D (0.69) HTR1DHTR1BHTR2AMEN1ALDH1A1
SCHEMBL8652262 0.84 HTR1D (0.68) HTR1DHTR1BHTR2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102535-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-09-29 EP disclosed
US-6399656-B1 USING A BENZOPYRAN-3-CARBOXAMIDE COMPOUND SMITHKLINE BEECHAM CORPORATION 2002-06-04 US disclosed
EP-1102535-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-05-30 EP disclosed
WO-2000006085-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed