SCHEMBL6604045

SCHEMBL6604045

COc1cc2c(cc1CNC1CCCN(C(=O)OC(C)(C)C)C1c1ccccc1)CCC(=S)N2C

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.44
HCRTR2 O43614 1/20 0.39
CFTR P13569 3/20 0.37
CYP2D6 P10635 4/20 0.37
KDM1A O60341 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7030797 1.00 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL6607867 0.97 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL8664244 0.92 TACR1 (0.45) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL6606866 0.92 TACR1 (0.45) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL6606522 0.87 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL7030644 0.87 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL7032701 0.86 TACR1 (0.46) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL6604119 0.86 TACR1 (0.46) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL6608982 0.84 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A
SCHEMBL7026966 0.84 TACR1 (0.44) TACR1HCRTR2CFTRCYP2D6KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175417-B1 SUBSTITUTED BENZOLACTAM COMPOUNDS PFIZER PROD INC (US) 2004-01-07 EP disclosed