SCHEMBL6604699

SCHEMBL6604699

COc1cc2c(cc1N1C[C@@H](C)N(C)[C@@H](C)C1)N(C(=O)Cc1cccc(F)c1F)CC2

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 18/20 0.84
HTR1D P28221 16/20 0.84
HTR1A P08908 4/20 0.66
GHSR Q92847 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604697 1.00 HTR1B (0.84) HTR1BHTR1DHTR1AGHSR
SCHEMBL6603215 0.91 HTR1B (1.00) HTR1BHTR1DHTR1AGHSR
SCHEMBL6603212 0.91 HTR1B (1.00) HTR1BHTR1DHTR1AGHSR
SCHEMBL6603524 0.91 HTR1B (0.79) HTR1BHTR1DHTR1AGHSR
SCHEMBL6606344 0.91 HTR1B (0.81) HTR1BHTR1DHTR1AGHSR
SCHEMBL6606346 0.91 HTR1B (0.81) HTR1BHTR1DHTR1AGHSR
SCHEMBL6603529 0.91 HTR1B (0.79) HTR1BHTR1DHTR1AGHSR
SCHEMBL6604234 0.90 HTR1B (1.00) HTR1BHTR1DHTR1AGHSR
SCHEMBL6604237 0.90 HTR1B (1.00) HTR1BHTR1DHTR1AGHSR
SCHEMBL6606649 0.90 HTR1B (1.00) HTR1BHTR1DHTR1AGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216239-B1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2004-02-11 EP claimed
EP-1216239-B1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2004-02-11 EP disclosed