SCHEMBL6609721

SCHEMBL6609721

O=C1CC(c2cccc(-c3nc(OC(=O)O)cs3)c2)=Nc2ccc(-c3ccccc3F)cc2N1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.53
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GRM2 Q14416 2/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5868974 0.88 CYP3A4 (0.55) CYP3A4GRM2RAB9ASMN1; SMN2
SCHEMBL5869071 0.85 CYP3A4 (0.56) CYP3A4GRM2RAB9ASMN1; SMN2
SCHEMBL5869000 0.83 CYP3A4 (0.51) CYP3A4NPC1GRM2RAB9ASMN1; SMN2
SCHEMBL5563880 0.78 CYP3A4 (0.69) CYP3A4GRM2
SCHEMBL5868932 0.76 GRM2 (0.50) CYP3A4GRM2RAB9ASMN1; SMN2
SCHEMBL2319292 0.76 CYP3A4 (0.66) CYP3A4RAB9ASMN1; SMN2
SCHEMBL5558069 0.75 CYP3A4 (0.66) CYP3A4GRM2
SCHEMBL5557822 0.75 GRM2 (0.69) CYP3A4GRM2
SCHEMBL5557011 0.75 CYP3A4 (0.65) CYP3A4GRM2RAB9ASMN1; SMN2
SCHEMBL6477792 0.75 CYP3A4 (0.65) CYP3A4GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224175-B1 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2004-03-17 EP claimed