SCHEMBL6610176

SCHEMBL6610176

CC(C)(C)OC(=O)C[C@H](NC(=O)OCc1ccccc1)C(O)COc1cccc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.53
SYK P43405 1/20 0.44
CYP2D6 P10635 4/20 0.43
ADRB2 P07550 4/20 0.41
ADRB1 P08588 4/20 0.41
SIGMAR1 Q99720 4/20 0.41
CYP1A2 P05177 3/20 0.41
SLC6A4 P31645 3/20 0.41
HTR2B P41595 3/20 0.41
NR2E1 Q9Y466 3/20 0.41
ALDH1A1 P00352 3/20 0.41
ADRB3 P13945 3/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
HTR6 P50406 3/20 0.41
SCN1A P35498 2/20 0.41
SLC10A1 Q14973 2/20 0.41
SCN2A Q99250 2/20 0.41
SCN3A Q9NY46 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6612201 0.85 SYK (0.49) CASP1SYKKLK5KLK7
SCHEMBL15095154 0.81 SYK (0.58) CASP1SYKKLK5
SCHEMBL7404713 0.81 SYK (0.53) CASP1SYKKLK5
SCHEMBL87318 0.81 SYK (0.58) CASP1SYKKLK5
SCHEMBL79132 0.80 SYK (0.44) SYKKLK5KLK7
SCHEMBL3213032 0.80 SYK (0.44) SYKKLK5KLK7
SCHEMBL79910 0.80 SYK (0.44) SYKKLK5KLK7
SCHEMBL7399633 0.79 SYK (0.47) SYKKLK5KLK7
SCHEMBL27885868 0.79 SYK (0.55) SYKKLK5
SCHEMBL27658167 0.79 SYK (0.55) SYKKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212309-B1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2004-08-18 EP disclosed
US-6747050-B1 INHIBITING THE ACTIVITY OF CASPASES, PREVENTING INFLAMMATION AND APOPTOSIS LG CHEM INVESTMENT LTD. (KR) 2004-06-08 US disclosed
EP-1212309-A4 CASPASE INHIBITOR LG CHEM INVESTMENT LTD (KR) 2002-11-27 EP disclosed
EP-1212309-A1 CASPASE INHIBITOR LG Chem Investment, Ltd. (KR) 2002-06-12 EP disclosed
WO-2001021600-A1 CASPASE INHIBITOR LG CHEM INVESTMENT LTD. (KR) 2001-03-29 WO disclosed