SCHEMBL6616489

SCHEMBL6616489

c1ccc(CC2CNc3ccccc3CN2)cc1

nearest known ligand 0.97

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.97
KMT2A Q03164 1/20 0.97
POLB P06746 1/20 0.42
PNMT P11086 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6618053 0.83 MEN1 (0.68) MEN1KMT2APOLBPNMT
SCHEMBL6614572 0.83 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6617044 0.83 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6616133 0.83 MEN1 (0.68) MEN1KMT2APOLBPNMT
SCHEMBL6613682 0.83 MEN1 (0.68) MEN1KMT2APOLBPNMT
SCHEMBL6615945 0.83 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6633687 0.83 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL6618257 0.82 MEN1 (0.68) MEN1KMT2APOLB
SCHEMBL10324241 0.80 MEN1 (0.65) MEN1KMT2APNMT
SCHEMBL5058983 0.80 MEN1 (0.65) MEN1KMT2APNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1481975-A1 Inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-01 EP disclosed
EP-0892797-A4 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL MYERS SQUIBB CO (US) 2004-10-20 EP disclosed
US-6455523-B1 ADMINISTERING 1,4-BENZODIAZEPINE DERIVATIVE AS ANTITUMOR OR ANTICARCINOGENIC AGENT BRISTOL-MYERS SQUIBB COMPANY 2002-09-24 US disclosed
US-6011029-A BENZODIAZEPINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-04 US disclosed
EP-0892797-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-01-27 EP disclosed
WO-1997030992-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1997-08-28 WO disclosed