SCHEMBL6619489

SCHEMBL6619489

CCOC(=O)CCCC1(NC(=O)c2cccs2)Nc2ccc(C(=O)N(C)C3CCCCC3)cc2N1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITK Q08881 12/20 0.55
ALDH1A1 P00352 4/20 0.36
ACKR3 P25106 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6619700 0.90 ITK (0.50) ITKALDH1A1ACKR3
SCHEMBL6621403 0.88 ITK (0.48) ITKACKR3
SCHEMBL6620631 0.88 ITK (0.48) ITKACKR3
SCHEMBL6620130 0.81 ITK (0.42) ITKALDH1A1
SCHEMBL6766640 0.73 ITK (0.92) ITK
SCHEMBL6619252 0.66 PTGER4 (0.48) ITKALDH1A1MAPT
SCHEMBL15562950 0.64 ITK (0.61) ITKALDH1A1ACKR3MAPTHTT
SCHEMBL6618857 0.64 MAPT (0.61) ITKALDH1A1LMNAMAPTHTT
SCHEMBL6771407 0.62 ITK (0.88) ITK
SCHEMBL31758152 0.62 KDM4E (0.60) ALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1448199-A1 BENZIMIDAZOLES USEFUL AS PROTEIN KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-08-25 EP disclosed
WO-2003041708-A1 BENZIMIDAZOLES USEFUL AS PROTEIN KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2003-05-22 WO disclosed