SCHEMBL6619862

SCHEMBL6619862

CS(=O)(=O)N1Cc2cc(Br)ccc2NCC1CCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 14/20 0.57
FNTB P49356 14/20 0.57
BRD4 O60885 1/20 0.36
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633343 0.89 FNTA (0.56) FNTAFNTBBRD4
SCHEMBL6614995 0.89 FNTA (0.56) FNTAFNTBBRD4
SCHEMBL6635226 0.82 FNTA (0.43) FNTAFNTBBRD4
SCHEMBL6614821 0.82 FNTA (0.41) FNTAFNTBBRD4KMT2A
SCHEMBL6619615 0.81 FNTA (0.52) FNTAFNTB
SCHEMBL6635340 0.81 FNTA (0.52) FNTAFNTB
SCHEMBL6619564 0.79 FNTA (0.60) FNTAFNTBKMT2A
SCHEMBL6616053 0.78 FNTA (0.45) FNTAFNTBBRD4KMT2A
SCHEMBL6616628 0.77 FNTA (0.40) FNTAFNTBBRD4
SCHEMBL6637318 0.76 FNTA (0.56) FNTAFNTBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1481975-A1 Inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-01 EP disclosed
EP-0892797-A4 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL MYERS SQUIBB CO (US) 2004-10-20 EP disclosed
US-6455523-B1 ADMINISTERING 1,4-BENZODIAZEPINE DERIVATIVE AS ANTITUMOR OR ANTICARCINOGENIC AGENT BRISTOL-MYERS SQUIBB COMPANY 2002-09-24 US disclosed
US-6011029-A BENZODIAZEPINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-01-04 US disclosed
EP-0892797-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-01-27 EP disclosed
WO-1997030992-A1 INHIBITORS OF FARNESYL PROTEIN TRANSFERASE BRISTOL-MYERS SQUIBB COMPANY (US) 1997-08-28 WO disclosed