SCHEMBL6620729

SCHEMBL6620729

CCC(C)Nc1cc2c(cc1C(F)(F)F)NC(=O)CC(c1cccc(-n3ccnn3)c1)=N2

nearest known ligand 0.80

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166900 0.89 CYP3A4 (0.55) CYP3A4
SCHEMBL6165499 0.84 CYP3A4 (0.55) CYP3A4
SCHEMBL6433551 0.84 CYP3A4 (0.67) CYP3A4
SCHEMBL6164338 0.83 CYP3A4 (0.60) CYP3A4
SCHEMBL6164688 0.83 CYP3A4 (0.56) CYP3A4
SCHEMBL6433608 0.83 GRM2 (0.70) CYP3A4
SCHEMBL6433387 0.82 CYP3A4 (0.62) CYP3A4
SCHEMBL6434645 0.82 GRM2 (0.73) CYP3A4
SCHEMBL6164415 0.78 CYP3A4 (0.55) CYP3A4
SCHEMBL6165350 0.75 CYP3A4 (0.55) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed