SCHEMBL6621603

SCHEMBL6621603

COc1cc(C(=O)O)ccc1OC(C)N(C)C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.65
CA1 P00915 2/20 0.65
CA2 P00918 2/20 0.65
CA4 P22748 2/20 0.65
CA6 P23280 2/20 0.65
CA7 P43166 2/20 0.65
CA9 Q16790 2/20 0.65
CA14 Q9ULX7 2/20 0.65
TPMT P51580 1/20 0.65
TSHR P16473 4/20 0.56
TTR P02766 2/20 0.54
HTT P42858 2/20 0.53
LMNA P02545 3/20 0.51
RAB9A P51151 2/20 0.51
MAPK1 P28482 1/20 0.51
NPSR1 Q6W5P4 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6619936 0.94 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL6622310 0.87 MAPT (0.59) CA12CA1CA2CA4CA6
SCHEMBL1015345 0.84 CA12 (0.73) CA12CA1CA2CA4CA6
SCHEMBL1554712 0.83 CA12 (0.71) CA12CA1CA2CA4CA6
Veratric Acid SCHEMBL114848 0.80 CA12 (1.00) CA12CA1CA2CA4CA6
Veratric Acid SCHEMBL29386353 0.80 CA12 (1.00) CA12CA1CA2CA4CA6
Veratric Acid SCHEMBL976032 0.80 CA12 (1.00) CA12CA1CA2CA4CA6
SCHEMBL2564619 0.80 CA12 (0.71) CA12CA1CA2CA4CA6
SCHEMBL22064771 0.79 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL18031240 0.79 CA12 (0.65) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067894-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-09-08 EP disclosed
US-6518267-B1 Protease inhibitors SMITHKLINE BEECHAM CORPORATION 2003-02-11 US disclosed
EP-1067894-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-01-17 EP disclosed
WO-1999059526-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO disclosed