SCHEMBL6622018

SCHEMBL6622018

OC(CCl)c1cc2ccccc2o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.56
HIF1A Q16665 1/20 0.56
KDM4E B2RXH2 2/20 0.43
FLT3 P36888 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
MGLL Q99685 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TYR P14679 1/20 0.42
DAO P14920 1/20 0.42
AKR1B1 P15121 1/20 0.42
HPGD P15428 1/20 0.42
AGXT P21549 1/20 0.40
MAOB P27338 4/20 0.39
CYP2A6 P11509 2/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TSHR P16473 2/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610235 1.00 CYP2D6 (0.56) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL6612005 1.00 CYP2D6 (0.56) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL29172969 0.81 CYP2D6 (0.60) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL8158785 0.81 CYP2D6 (0.56) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL24173635 0.81 CYP2D6 (0.60) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL28594760 0.80 CYP2D6 (0.44) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL6610233 0.77 CYP2D6 (0.60) CYP2D6HIF1AKDM4EHSD17B10TDP1
SCHEMBL6284878 0.77 CYP2D6 (0.56) CYP2D6HIF1AKDM4EFLT3LOXL2
SCHEMBL6608279 0.77 CYP2D6 (0.60) CYP2D6HIF1AKDM4EHSD17B10TDP1
SCHEMBL23239223 0.77 CYP2D6 (0.52) CYP2D6HIF1AKDM4EFLT3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458719-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2004-09-22 EP disclosed
WO-2003053971-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2003-07-03 WO disclosed