SCHEMBL6626074

SCHEMBL6626074

C[C@@H]1OCCN(c2nc(N3CCOCC3)cc(-n3cnc4ccccc43)n2)[C@H]1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 3/20 0.53
HRH4 Q9H3N8 1/20 0.50
LCK P06239 1/20 0.49
PDCD1 Q15116 6/20 0.49
CD274 Q9NZQ7 6/20 0.49
ATR Q13535 5/20 0.49
CHEK1 O14757 4/20 0.49
ATRIP Q8WXE1 4/20 0.49
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 2/20 0.44
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PIK3CD O00329 1/20 0.41
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6626063 1.00 PIK3CB (0.53) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625589 1.00 PIK3CB (0.53) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625592 1.00 PIK3CB (0.53) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625597 1.00 PIK3CB (0.53) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6626388 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6626384 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625790 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL5213834 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL6625795 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274
SCHEMBL5213821 0.94 PIK3CB (0.58) PIK3CBHRH4LCKPDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020462-B1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KK (JP) 2004-02-11 EP disclosed
US-6251900-B1 Heterocyclic compounds and antitumor agent containing the same as active ingredient ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2001-06-26 US disclosed
EP-1020462-A1 HETEROCYCLIC COMPOUNDS AND ANTITUMOR AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-07-19 EP disclosed