SCHEMBL6626769

SCHEMBL6626769

Cc1cc(F)ccc1C1CC(N2CCN(C)CC2=O)CCN1C(=O)NC[C@H](C)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.56
SIGMAR1 Q99720 2/20 0.56
PTAFR P25105 1/20 0.56
CYP3A4 P08684 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600387 0.87 TACR1 (0.57) TACR1SIGMAR1PTAFRCYP3A4
SCHEMBL6626766 0.85 TACR1 (0.76) TACR1SIGMAR1PTAFRCYP3A4
SCHEMBL3228336 0.80 TACR1 (0.54) TACR1SIGMAR1PTAFRCYP3A4
SCHEMBL4398271 0.79 TACR1 (0.54) TACR1SIGMAR1CYP3A4
SCHEMBL5618540 0.79 TACR1 (0.47) TACR1SIGMAR1PTAFRCYP3A4
SCHEMBL6365455 0.79 TACR1 (0.47) TACR1SIGMAR1PTAFRCYP3A4
SCHEMBL5618542 0.79 TACR1 (0.47) TACR1SIGMAR1PTAFRCYP3A4
Hydrochloric Acid SCHEMBL5619955 0.77 TACR1 (0.55) TACR1SIGMAR1PTAFRCYP3A4
Hydrochloric Acid SCHEMBL6623896 0.77 TACR1 (0.55) TACR1SIGMAR1PTAFRCYP3A4
Hydrochloric Acid SCHEMBL5619491 0.77 TACR1 (0.55) TACR1SIGMAR1PTAFRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472243-A1 PIPERIDINE DERIVATIVES AND THEIR USE AS ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 2004-11-03 EP claimed
WO-2003066621-A1 PIPERIDINE DERIVATIVES AND THEIR USE AS ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 2003-08-14 WO claimed