SCHEMBL6635013

SCHEMBL6635013

CCCC(=O)Nc1cnccc1-c1ccccc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 1/20 0.48
MAPK1 P28482 1/20 0.48
KDM6B O15054 2/20 0.45
KDM4D Q6B0I6 2/20 0.45
KDM4C Q9H3R0 2/20 0.45
EGLN3 Q9H6Z9 1/20 0.45
F2R P25116 1/20 0.45
ALDH1A1 P00352 2/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
TP53 P04637 2/20 0.44
NOTUM Q6P988 1/20 0.44
POLB P06746 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635289 0.89 PARP14 (0.45) PARP14MAPK1KDM6BKDM4DKDM4C
SCHEMBL16628650 0.83 GPBAR1 (0.47) KDM4DKDM4C
SCHEMBL5768636 0.79 MAPK1 (0.49) MAPK1KDM6BKDM4DKDM4CEGLN3
SCHEMBL6635011 0.78 MAPT (0.51) RAB9ASMN1; SMN2TP53NOTUMMAPT
SCHEMBL6637207 0.78 TSHR (0.48) RAB9ASMN1; SMN2TP53MAPTAAK1
SCHEMBL12097325 0.75 NAMPT (0.44) RAB9A
SCHEMBL6658490 0.75 MAPK1 (0.69) MAPK1ALDH1A1RAB9ASMN1; SMN2POLB
SCHEMBL6634845 0.74 CYP1A2 (0.50) MAPK1KDM4CALDH1A1LIMK1
SCHEMBL2003108 0.72 KDM4C (0.45) KDM4CLIMK1
SCHEMBL21258161 0.72 ATR (0.45) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035115-B1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists HOFFMANN LA ROCHE (CH) 2004-09-29 EP claimed