SCHEMBL6635592

SCHEMBL6635592

CCOC(=O)CN(c1ccc2c(c1)cc(CNc1ccc(C(=N)N)cc1)n2C)S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F2 P00734 9/20 0.66
NQO2 P16083 2/20 0.45
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
SLC22A2 O15244 1/20 0.37
F10 P00742 1/20 0.37
PLG P00747 1/20 0.37
PLAT P00750 1/20 0.37
PROC P04070 1/20 0.37
HPN P05981 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
SLC47A2 Q86VL8 1/20 0.37
SLC47A1 Q96FL8 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.36
TP53 P04637 2/20 0.36
PKLR P30613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635710 0.91 F2 (0.78) F2NQO2SLC22A2F10PLG
SCHEMBL8031709 0.90 F2 (0.64) F2NQO2GAATSHRF10
SCHEMBL6635963 0.89 F2 (0.65) F2NQO2GAATSHRF10
Hydrochloric Acid SCHEMBL8028886 0.89 F2 (0.64) F2NQO2GAATSHRF10
SCHEMBL6640290 0.89 F2 (0.83) F2NQO2SLC22A2F10PLG
SCHEMBL6635063 0.88 F2 (0.51) F2GAATSHRALDH1A1MAPT
Hydrochloric Acid SCHEMBL8016067 0.84 F2 (0.66) F2NQO2GAATSHRSLC22A2
Hydrochloric Acid SCHEMBL8026688 0.84 F2 (0.59) F2NQO2GAATSHRF10
SCHEMBL8130727 0.84 F2 (0.54) F2GAATSHRALDH1A1MAPT
SCHEMBL6635608 0.83 F2 (0.81) F2NQO2SLC22A2F10PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed