SCHEMBL6637263

SCHEMBL6637263

CC(NC(=O)OC(C)(C)C)C(O)CN

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.51
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA7 P43166 2/20 0.49
CTSK P43235 11/20 0.43
CTSS P25774 6/20 0.42
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17282912 1.00 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL14384109 1.00 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL6623815 1.00 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL14384110 1.00 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL3380313 0.84 CYP2D6 (0.53) CYP2D6CA1CA2CA7CTSK
SCHEMBL31606449 0.84 CYP2D6 (0.53) CYP2D6CA1CA2CA7CTSK
SCHEMBL14931110 0.84 CYP2D6 (0.53) CYP2D6CA1CA2CA7CTSK
SCHEMBL18359144 0.84 CA1 (0.50) CYP2D6CA1CA2CA7CTSK
SCHEMBL13538162 0.84 CYP2D6 (0.53) CYP2D6CA1CA2CA7CTSK
SCHEMBL14923535 0.82 CA1 (0.53) CYP2D6CA1CA2CA7CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067894-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-09-08 EP disclosed
EP-1067894-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-01-17 EP disclosed
WO-1999059526-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO disclosed