SCHEMBL6637608

SCHEMBL6637608

CC(=O)NCCNc1nc(Nc2ccc(C(=O)NCCc3ccccc3)cc2)ncc1C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 18/20 0.60
CHEK1 O14757 1/20 0.59
FLT3 P36888 1/20 0.59
JAK2 O60674 1/20 0.54
NTRK1 P04629 1/20 0.54
TYK2 P29597 1/20 0.54
KDR P35968 1/20 0.54
JAK3 P52333 1/20 0.54
PTK2B Q14289 1/20 0.54
NTRK3 Q16288 1/20 0.54
NTRK2 Q16620 1/20 0.54
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1916872 0.87 FLT3 (0.60) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL3283893 0.87 CHEK1 (0.63) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL1917544 0.86 PTK2 (0.71) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL1916885 0.86 CHEK1 (0.68) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL6639386 0.85 CYP3A4 (0.52) PTK2CHEK1FLT3GSK3AGSK3B
SCHEMBL1917639 0.84 PTK2 (0.66) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL1916946 0.84 CHEK1 (0.57) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL1919207 0.84 CHEK1 (0.57) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL3284837 0.84 PTK2 (0.62) PTK2CHEK1FLT3JAK2NTRK1
SCHEMBL3291976 0.83 PTK2 (0.61) PTK2CHEK1FLT3JAK2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1438053-A1 PYRIMIDINE DERIVATIVES, PHARMACEUTICAL AGENT CONTAINING SAID COMPOUNDS, USE AND METHOD FOR MAKING SAME Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-07-21 EP disclosed
WO-2003032997-A1 PYRIMIDINE DERIVATIVES, PHARMACEUTICAL AGENT CONTAINING SAID COMPOUNDS, USE AND METHOD FOR MAKING SAME BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-04-24 WO disclosed