SCHEMBL6638686

SCHEMBL6638686

CCOC(=O)CN(c1ccc2c(C)c(CNc3ccc(C#N)cc3)oc2c1)S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.44
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
PKM P14618 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
TP53 P04637 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8032187 0.90 F2 (0.42) F2GAATSHRPKMALDH1A1
SCHEMBL6637732 0.89 F2 (0.43) F2GAATSHRPKMALDH1A1
SCHEMBL6636555 0.89 F2 (0.58) F2GAATSHRPKMALDH1A1
Hydrochloric Acid SCHEMBL6636009 0.88 F2 (0.57) F2GAATSHRPKMALDH1A1
SCHEMBL6636960 0.85 F2 (0.41) F2GAAPKMALDH1A1MAPT
SCHEMBL6636557 0.85 F2 (0.46) F2GAATSHRALDH1A1MAPT
SCHEMBL8030596 0.84 F2 (0.41) F2GAATSHRPKMALDH1A1
SCHEMBL6638864 0.84 HCRTR2 (0.43) TSHRALDH1A1MAPTLMNA
SCHEMBL6635830 0.83 HCRTR2 (0.32) F2ALDH1A1MAPTLMNA
SCHEMBL6634473 0.83 F2 (0.39) F2PKMALDH1A1MAPTFNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed