SCHEMBL6640458

SCHEMBL6640458

Cn1c(COc2cccc(C(=N)N)c2)nc2cc(NS(=O)(=O)c3cccc4cccnc34)ccc21

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
F2 P00734 12/20 0.74
FABP1 P07148 1/20 0.46
ALDH1A1 P00352 2/20 0.46
TP53 P04637 1/20 0.46
HTT P42858 1/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.45
ST14 Q9Y5Y6 1/20 0.44
BRD4 O60885 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638828 0.86 F2 (0.58) F2FABP1ALDH1A1TP53HTT
SCHEMBL6639365 0.85 F2 (0.68) F2ALDH1A1PKM
Hydrochloric Acid SCHEMBL8032926 0.84 F2 (0.98) F2ALDH1A1PKMST14BRD4
SCHEMBL6635570 0.83 F2 (0.79) F2ALDH1A1PKMST14BRD4
SCHEMBL6636479 0.81 F2 (0.64) F2FABP1ALDH1A1ST14
Hydrochloric Acid SCHEMBL8031754 0.80 F2 (0.75) F2ALDH1A1GAAPKMST14
SCHEMBL6640826 0.80 F2 (0.63) F2FABP1ALDH1A1ST14
SCHEMBL6637955 0.80 F2 (0.62) F2FABP1ALDH1A1TP53HTT
SCHEMBL6638878 0.79 F2 (0.78) F2ALDH1A1PKMST14BRD4
SCHEMBL6637221 0.79 F2 (0.61) F2FABP1ALDH1A1ST14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100795-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES HAVING, IN PARTICULAR, A THROMBIN INHIBITIVE EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2004-06-09 EP disclosed
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed