SCHEMBL6640562

SCHEMBL6640562

CCCc1c(Br)n(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(CCCF)CC4)ccc3OCC)nc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.63
PDE3B Q13370 3/20 0.63
PDE3A Q14432 3/20 0.63
HDAC1 Q13547 2/20 0.62
HDAC6 Q9UBN7 2/20 0.62
HDAC2 Q92769 1/20 0.62
PDE1A P54750 2/20 0.60
PDE1B Q01064 2/20 0.60
PDE1C Q14123 2/20 0.60
PDE2A O00408 1/20 0.60
ABCC4 O15439 1/20 0.60
ABCC5 O15440 1/20 0.60
PDE6D O43924 1/20 0.60
PDE8A O60658 1/20 0.60
PDE9A O76083 1/20 0.60
ABCB11 O95342 1/20 0.60
CYP3A4 P08684 1/20 0.60
HTR1A P08908 1/20 0.60
PDE6A P16499 1/20 0.60
PDE6G P18545 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6643883 0.96 PDE5A (0.65) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6643001 0.93 PDE5A (0.69) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6643348 0.91 PDE5A (0.63) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6643219 0.91 PDE5A (0.63) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6642850 0.91 PDE5A (0.75) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6640125 0.91 PDE5A (0.66) PDE5A
SCHEMBL6645339 0.90 PDE5A (0.73) PDE5APDE3BPDE3APDE1APDE1B
SCHEMBL6485807 0.88 PDE5A (0.81) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL6643613 0.87 PDE5A (0.65) PDE5APDE3BPDE3AHDAC1HDAC6
Hydrochloric Acid SCHEMBL6643166 0.87 PDE5A (0.80) PDE5APDE3BPDE3AHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257553-B1 PYRROLOPYRIMIDINONE DERIVATIVES, PROCESS OF PREPARATION AND USE SK CHEMICALS CO LTD (KR) 2004-05-26 EP disclosed