SCHEMBL6644162

SCHEMBL6644162

COC(=O)c1ccc(-c2cc[nH]c(=O)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
NOTUM Q6P988 1/20 0.51
ERN1 O75460 1/20 0.50
CA1 P00915 5/20 0.47
CA2 P00918 5/20 0.47
CA12 O43570 4/20 0.47
CA9 Q16790 4/20 0.47
CA14 Q9ULX7 3/20 0.47
ALDH2 P05091 4/20 0.47
TDP1 Q9NUW8 1/20 0.46
CA7 P43166 1/20 0.46
SETD7 Q8WTS6 1/20 0.45
POLB P06746 1/20 0.44
PTPN1 P18031 1/20 0.44
CDK8 P49336 1/20 0.44
PLAU P00749 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9950445 0.86 CDK8 (0.59) EGFRNOTUMERN1CA1CA2
SCHEMBL205408 0.81 CA1 (0.48) KDM4EALDH1A1CA1CA2CA12
SCHEMBL6638344 0.80 NOTUM (0.63) EGFRKDM4EALDH1A1NOTUMERN1
SCHEMBL19387238 0.78 CA1 (0.70) EGFRKDM4EALDH1A1ERN1CA1
Biphenyl Dimethyl Dicarboxylate SCHEMBL68521 0.78 CA1 (0.70) EGFRKDM4EALDH1A1ERN1CA1
SCHEMBL7853544 0.78 CA1 (0.50) KDM4EALDH1A1CA1CA2CA12
SCHEMBL16749655 0.77 CA1 (0.58) EGFRKDM4EALDH1A1ERN1CA1
SCHEMBL10009170 0.77 CA1 (0.61) EGFRKDM4EALDH1A1ERN1CA1
SCHEMBL16749645 0.77 CA1 (0.61) EGFRKDM4EALDH1A1ERN1CA1
Biphenyl Dimethyl Dicarboxylate SCHEMBL2890577 0.76 CA1 (0.67) EGFRKDM4EALDH1A1ERN1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931060-A4 SUBSTITUTED N- (AMINOIMINOMETHYL OR AMINOMETHYL)PHENYL]PROPYL AMIDES AVENTIS PHARMA INC (US) 2004-10-06 EP disclosed
EP-0931060-A1 SUBSTITUTED N- (AMINOIMINOMETHYL OR AMINOMETHYL)PHENYL]PROPYL AMIDES RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-07-28 EP disclosed
WO-1999000356-A1 SUBSTITUTED N-[(AMINOIMINOMETHYL OR AMINOMETHYL)PHENYL]PROPYL AMIDES RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1999-01-07 WO disclosed