SCHEMBL6645381

SCHEMBL6645381

CO[C@@H](CN1CC(C)(C)Cn2c1nc(-c1ccncn1)cc2=O)c1ccccc1.COc1ccccc1C(CN1CC(C)(C)Cn2c1nc(-c1ccncn1)cc2=O)OC

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.43
CYP2D6 P10635 6/20 0.43
CYP1A2 P05177 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3572812 0.97 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3570581 0.93 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3570578 0.93 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3570579 0.93 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3576221 0.90 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3561620 0.90 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3563256 0.88 GSK3B (0.39) GSK3BCYP2D6CYP1A2
SCHEMBL3576425 0.87 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3571964 0.85 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3566135 0.85 GSK3B (0.41) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430056-A1 SUBSTITUTED 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIMIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES FOR NEURODEGENERATIVE DISORDERS Sanofi-Aventis (FR) 2004-06-23 EP claimed
WO-2003027115-A1 SUBSTITUTED 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIMIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES FOR NEURODEGENERATIVE DISORDERS SANOFI-SYNTHELABO (FR) 2003-04-03 WO claimed