SCHEMBL6645979

SCHEMBL6645979

CC1(C)CN(CC(=O)c2ccccc2)c2nc(-c3ccncc3)c(F)c(=O)n2C1.O=c1cc(-c2ccncc2)nc2n1CC(F)(F)CN2C[C@@H](O)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 10/20 0.37
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6645977 1.00 GSK3B (0.37) GSK3BPIK3R1PIK3CAADORA2AADORA1
SCHEMBL4872302 0.84 GSK3B (0.35) GSK3B
SCHEMBL4870914 0.84 GSK3B (0.37) GSK3BPIK3R1PIK3CA
SCHEMBL4870926 0.84 GSK3B (0.37) GSK3BPIK3R1PIK3CA
SCHEMBL4870920 0.84 GSK3B (0.37) GSK3BPIK3R1PIK3CA
Hydrochloric Acid SCHEMBL4869542 0.83 GSK3B (0.35) GSK3B
SCHEMBL6675120 0.83 GSK3B (0.46) GSK3BPIK3R1PIK3CAADORA1
SCHEMBL6675118 0.83 GSK3B (0.46) GSK3BPIK3R1PIK3CAADORA1
SCHEMBL4865736 0.82 GSK3B (0.48) GSK3BPIK3R1PIK3CA
SCHEMBL4870991 0.82 GSK3B (0.51) GSK3BPIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430057-A2 SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO 1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO 1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES Sanofi-Aventis (FR) 2004-06-23 EP claimed
WO-2003027116-A2 SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES SANOFI-SYNTHELABO (FR) 2003-04-03 WO claimed