SCHEMBL6648271

SCHEMBL6648271

COc1cc(F)ccc1C(=O)CN1CC(C)(C)Cn2c1nc(-c1ccncn1)cc2=O.COc1cc(F)ccc1C(O)CN1CC(C)(C)Cn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.44
CYP2D6 P10635 5/20 0.42
CYP1A2 P05177 3/20 0.40
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3573673 0.93 GSK3B (0.46) GSK3BCYP2D6CYP1A2PIK3R1PIK3CA
SCHEMBL3565488 0.92 GSK3B (0.49) GSK3BCYP2D6CYP1A2
SCHEMBL6669743 0.86 GSK3B (0.38) GSK3BCYP2D6CYP1A2
SCHEMBL3576425 0.86 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3576221 0.84 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3571557 0.84 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3575938 0.81 GSK3B (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL3568067 0.80 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL3571249 0.80 GSK3B (0.44) GSK3BCYP2D6CYP1A2
SCHEMBL3572812 0.78 GSK3B (0.45) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430056-A1 SUBSTITUTED 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIMIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES FOR NEURODEGENERATIVE DISORDERS Sanofi-Aventis (FR) 2004-06-23 EP claimed
WO-2003027115-A1 SUBSTITUTED 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIMIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES FOR NEURODEGENERATIVE DISORDERS SANOFI-SYNTHELABO (FR) 2003-04-03 WO claimed