SCHEMBL6652492

SCHEMBL6652492

COc1ccnc(N2CCN(C(=O)c3sccc3F)CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.47
HCRTR2 O43614 10/20 0.47
ALDH1A1 P00352 5/20 0.44
SLC6A7 Q99884 1/20 0.44
HPGD P15428 1/20 0.44
KDM4E B2RXH2 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PARP1 P09874 1/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7713964 0.99 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hypochlorous Acid SCHEMBL7713970 0.98 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
SCHEMBL6650527 0.88 HCRTR1 (0.49) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
SCHEMBL6649976 0.88 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
SCHEMBL6652566 0.87 HCRTR1 (0.45) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hydrochloric Acid SCHEMBL27484703 0.87 HCRTR1 (0.45) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hydrochloric Acid SCHEMBL6650987 0.87 HCRTR1 (0.48) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hydrochloric Acid SCHEMBL6652387 0.86 HCRTR1 (0.44) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hypochlorous Acid SCHEMBL6652392 0.86 HCRTR1 (0.44) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD
Hypochlorous Acid SCHEMBL6650991 0.86 HCRTR1 (0.48) HCRTR1HCRTR2ALDH1A1SLC6A7HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006110-B1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS ESTEVE LABOR DR (ES) 2004-02-11 EP claimed
US-6372746-B1 ANTICONVULSIVE AGENTS, SEDATIVES AND EATING DISORDERS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2002-04-16 US claimed
EP-1006110-A1 DERIVATIVES OF ACYL-PIPERAZINIL-PYRIMIDINS, PREPARATION THEREOF AND APPLICATION AS MEDICAMENTS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2000-06-07 EP claimed