SCHEMBL6661698

SCHEMBL6661698

Oc1ccc(Nc2cncc(Cl)n2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.69
BRAF P15056 4/20 0.56
GAA P10253 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
AURKA O14965 4/20 0.45
SCN5A Q14524 2/20 0.44
SCN9A Q15858 2/20 0.44
KCNH2 Q12809 1/20 0.44
GRM4 Q14833 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TNIK Q9UKE5 1/20 0.39
DHFR P00374 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2885798 0.85 CDK2 (0.73) CDK2BRAFSCN5ASCN9AKCNH2
SCHEMBL6302354 0.82 CDK2 (0.69) CDK2BRAFGAAMEN1KMT2A
SCHEMBL1678613 0.81 CDK2 (1.00) CDK2BRAFMEN1KMT2ASCN5A
SCHEMBL2932811 0.80 CDK2 (0.66) CDK2BRAFGAAKMT2ASMN1; SMN2
SCHEMBL6662179 0.80 CDK2 (0.66) CDK2BRAFMEN1KMT2APOLB
SCHEMBL1122444 0.79 CDK2 (0.65) CDK2BRAFGAAMEN1KMT2A
SCHEMBL6656588 0.79 BRAF (0.62) CDK2BRAFSMN1; SMN2POLBMAPT
SCHEMBL16739547 0.78 CDK2 (0.63) CDK2BRAFSCN5ASCN9AKCNH2
SCHEMBL6659290 0.76 CDK2 (1.00) CDK2MEN1KMT2A
SCHEMBL6662729 0.74 CDK2 (0.72) CDK2BRAFMEN1KMT2AGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004004730-A2 2-AMINOPYRAZINE DERIVATIVES AS INHIBITORS OF CYCLIN DEPENDENT KINASES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO claimed
WO-2004004730-A2 2-AMINOPYRAZINE DERIVATIVES AS INHIBITORS OF CYCLIN DEPENDENT KINASES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS ASTEX TECHNOLOGY LIMITED (GB) 2004-01-15 WO disclosed