SCHEMBL6663690

SCHEMBL6663690

C#CCN(CC#C)S(=O)(=O)c1ccc(-n2ncc3ccc4[nH]ncc4c32)cc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21067935 0.79 CA1 (0.54) CA12CA1CA2CA9
SCHEMBL5230987 0.79 CCNA2 (0.42)
SCHEMBL12886452 0.69 CCNA2 (0.37)
SCHEMBL5231014 0.64 CCNA2 (0.62)
SCHEMBL5232593 0.63 CCNA2 (0.74)
SCHEMBL10653112 0.62 TLR9 (0.39)
SCHEMBL1082207 0.61 GLA (0.69) CA12CA9
SCHEMBL5225835 0.60 CCNA2 (0.57)
SCHEMBL5228506 0.59 CCNA2 (0.46)
SCHEMBL13913086 0.59 CA1 (0.47) CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478357-A2 TRICYCLIC PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS Pharmacia Italia S.p.A. (IT) 2004-11-24 EP claimed
WO-2003070236-A2 TRICYCLIC PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA S.P.A. (IT) 2003-08-28 WO claimed