SCHEMBL6663910

SCHEMBL6663910

Cc1ccc2ncnc(Nc3cccc(C#N)c3)c2c1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.73
HTT P42858 3/20 0.67
MAPK1 P28482 2/20 0.67
KDM4E B2RXH2 1/20 0.67
EGFR P00533 8/20 0.67
ERBB2 P04626 2/20 0.62
MAPT P10636 2/20 0.61
LMNA P02545 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
HPGD P15428 2/20 0.60
F9 P00740 1/20 0.60
ALDH1A1 P00352 1/20 0.60
TP53 P04637 1/20 0.58
HIF1A Q16665 1/20 0.57
NCOA1 Q15788 1/20 0.55
NCOA3 Q9Y6Q9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27529543 0.88 EGFR (0.69) ABCG2HTTMAPK1KDM4EEGFR
Hydrochloric Acid SCHEMBL1507507 0.86 EGFR (0.67) ABCG2HTTMAPK1KDM4EEGFR
SCHEMBL8871863 0.85 EGFR (0.82) HTTMAPK1KDM4EEGFRERBB2
SCHEMBL1507715 0.84 ABCG2 (0.71) ABCG2EGFRERBB2MAPTLMNA
Hydrochloric Acid SCHEMBL9017046 0.83 ABCG2 (0.97) ABCG2HTTEGFRERBB2LMNA
SCHEMBL2101381 0.81 HTT (1.00) ABCG2HTTMAPK1KDM4EEGFR
SCHEMBL5565226 0.81 HTT (0.72) ABCG2HTTMAPK1KDM4EEGFR
SCHEMBL4741685 0.81 EGFR (0.80) HTTMAPK1KDM4EEGFRERBB2
SCHEMBL5569022 0.81 HTT (0.72) HTTMAPK1KDM4EEGFRERBB2
SCHEMBL5564456 0.81 MAPK1 (0.82) ABCG2HTTMAPK1KDM4EEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004013091-A2 4-ANILIDO SUBSTITUTED QUINAZOLINES AND USE THEREOF AS INHIBITORS OF EPIDERMAL GROWTH FACTOR RECEPTOR KINASES YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2004-02-12 WO disclosed