SCHEMBL6668568

SCHEMBL6668568

Cc1ccnc(NCCCC(=O)NCC(=O)NC(CC(=O)O)c2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.81

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 17/20 0.81
ITGB3 P05106 16/20 0.81
ITGB6 P18564 8/20 0.81
ITGB5 P18084 7/20 0.81
ITGA2B P08514 6/20 0.81
ITGB1 P05556 1/20 0.74
ITGA5 P08648 1/20 0.74
RAB9A P51151 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7170078 0.99 ITGAV (0.79) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7170092 0.99 ITGAV (0.79) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6670827 0.97 ITGAV (0.79) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7172733 0.96 ITGAV (0.77) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7172749 0.96 ITGAV (0.77) ITGAVITGB3ITGB6ITGB5ITGA2B
Trifluoroacetic Acid SCHEMBL6670246 0.95 ITGAV (0.82) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7204210 0.94 ITGAV (0.74) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6671946 0.93 ITGAV (0.79) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6671127 0.93 ITGAV (0.73) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7174477 0.93 ITGAV (0.78) ITGAVITGB3ITGB6ITGB5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP claimed
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US claimed
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US disclosed
EP-1153014-A2 BETA-ALANINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-11-14 EP disclosed
WO-2000048996-A2 β-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-08-24 WO disclosed