SCHEMBL6668614

SCHEMBL6668614

c1ccc(-c2cn3ccnc3s2)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.55
NPC1 O15118 6/20 0.55
RAB9A P51151 5/20 0.55
MAPT P10636 4/20 0.55
GLA P06280 2/20 0.55
POLB P06746 2/20 0.46
GAA P10253 1/20 0.46
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
LMNA P02545 4/20 0.43
CCR1 P32246 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL567444 0.79 EGFR (0.47) KDM4EGLAHDAC1HDAC2ALDH1A1
SCHEMBL3069800 0.72 KDM4E (1.00) KDM4ENPC1RAB9AMAPTGLA
SCHEMBL30326993 0.72 KDM4E (0.50) KDM4ENPC1RAB9AMAPTGLA
SCHEMBL28857293 0.71 KDM4E (0.95) KDM4ENPC1RAB9AMAPTGLA
SCHEMBL3085667 0.69 FLT3 (0.38) KDM4ENPC1RAB9ACYP1A2TP53
Dipyridyl SCHEMBL722577 0.67 KDM4E (0.93) KDM4ENPC1RAB9AMAPTGLA
Dipyridyl SCHEMBL3796795 0.67 KDM4E (0.93) KDM4ENPC1RAB9AMAPTGLA
Dipyridyl SCHEMBL29467582 0.67 KDM4E (0.93) KDM4ENPC1RAB9AMAPTGLA
Dipyridyl SCHEMBL721272 0.67 KDM4E (0.93) KDM4ENPC1RAB9AMAPTGLA
SCHEMBL146382 0.66 KDM4E (0.75) KDM4ENPC1RAB9AMAPTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185521-B1 SUBSTITUTED 1-AZA-2-IMINO-HETEROCYCLES AND THEIR USE AS ACTIVATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS DAIICHI SUNTORY PHARMA CO LTD (JP) 2004-10-06 EP disclosed