SCHEMBL6669229

SCHEMBL6669229

CC1(C)CCSc2ccc(C#Cc3ccc(C(=O)O)s3)cc21

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RARB P10826 16/20 0.61
RARG P13631 16/20 0.61
RARA P10276 14/20 0.61
CYP3A4 P08684 3/20 0.61
CYP26A1 O43174 2/20 0.61
KMT2A Q03164 1/20 0.51
RXRA P19793 6/20 0.47
CRABP2 P29373 1/20 0.46
RXRB P28702 4/20 0.41
RXRG P48443 4/20 0.41
SSTR5 P35346 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180433 0.86 RARB (0.64) RARBRARGRARACYP3A4CYP26A1
SCHEMBL30374339 0.86 RARB (0.64) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6667766 0.84 RARB (0.54) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9817648 0.83 CYP3A4 (0.76) RARBRARGRARACYP3A4CYP26A1
SCHEMBL19034088 0.82 RARB (0.62) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6052691 0.81 RARB (0.56) RARBRARGRARACYP3A4CYP26A1
SCHEMBL19342986 0.80 RARB (0.62) RARBRARGRARACYP3A4CYP26A1
SCHEMBL19342905 0.79 RARB (0.61) RARBRARGRARACYP3A4CYP26A1
SCHEMBL19342965 0.79 RARB (0.61) RARBRARGRARACYP3A4CYP26A1
SCHEMBL22198842 0.79 CYP3A4 (0.70) RARBRARGRARACYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-B1 USE OF DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN INC (US) 2004-09-08 EP claimed