SCHEMBL6670180

SCHEMBL6670180

COC(=O)CC(NC(=O)CNC(=O)CCCNc1ncccn1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 15/20 0.64
ITGB3 P05106 14/20 0.64
ITGB6 P18564 6/20 0.64
ITGB5 P18084 5/20 0.64
ITGA2B P08514 5/20 0.64
ITGB1 P05556 1/20 0.48
ITGA5 P08648 1/20 0.48
TACR3 P29371 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TAOK1 Q7L7X3 1/20 0.38
TAOK3 Q9H2K8 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ITGB8 P26012 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6670290 0.97 ITGAV (0.68) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6667525 0.91 ITGAV (0.78) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6669034 0.90 ITGAV (0.77) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7171385 0.89 ITGAV (0.76) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6668031 0.88 ITGAV (0.83) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7173522 0.88 ITGAV (0.59) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7171394 0.88 ITGAV (0.65) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6669430 0.87 ITGAV (0.82) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7173311 0.87 ITGAV (0.81) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6669087 0.86 ITGAV (0.70) ITGAVITGB3ITGB6ITGB5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153014-B1 BETA-ALANINE DERIVATIVES MERCK PATENT GMBH (DE) 2004-09-22 EP disclosed
US-6576637-B1 Such as 3-(4-methyl-3-nitrophenyl)-3-(2-(4-(pyridin-2-yl-amino)butyryl amino)acetylamino)propionic acid; thrombosis, heart infarct, coronary heart diseases, arteriosclerosis, inflammations, MERCK PATENT GMBH (DE) 2003-06-10 US disclosed