SCHEMBL6671573

SCHEMBL6671573

NCCCN.O=C(N[C@@H](CCCNCc1ccccn1)C(=O)O)c1ccc(CNCc2ccccn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.51
FOLH1 Q04609 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
FPGS Q05932 6/20 0.42
CHRM2 P08172 1/20 0.42
DHFR P00374 3/20 0.42
GRIA1 P42261 2/20 0.41
GPR132 Q9UNW8 1/20 0.41
HDAC1 Q13547 1/20 0.41
ERAP2 Q6P179 1/20 0.41
LNPEP Q9UIQ6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27566287 0.95 CXCR4 (0.53) CXCR4FOLH1NPC1LMNAPOLB
SCHEMBL6018116 0.95 CXCR4 (0.53) CXCR4FOLH1NPC1LMNAPOLB
Phenylhydrazine SCHEMBL6690774 0.91 CXCR4 (0.50) CXCR4FOLH1NPC1LMNAPOLB
SCHEMBL27568576 0.90 CXCR4 (0.47) CXCR4FOLH1KMT2AITGB3ITGA2B
SCHEMBL6667469 0.90 CXCR4 (0.47) CXCR4FOLH1KMT2AITGB3ITGA2B
SCHEMBL6018220 0.90 CXCR4 (0.51) CXCR4FOLH1NPC1LMNAPOLB
SCHEMBL6670076 0.90 CXCR4 (0.48) CXCR4FOLH1NPC1LMNAPOLB
SCHEMBL27616554 0.89 CXCR4 (0.54) CXCR4NPC1LMNAPOLBRAB9A
SCHEMBL6018126 0.89 CXCR4 (0.54) CXCR4NPC1LMNAPOLBRAB9A
SCHEMBL6018262 0.87 CXCR4 (0.57) CXCR4FOLH1NPC1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 CXCR4 1/4885FOLH1 2694/4885NPC1 943/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.