SCHEMBL6672263

SCHEMBL6672263

Cc1c(N2CC(F)C(C(O)CO)C2)c(F)cc2c(=O)[nH]c(=O)n(C3CC3)c12

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.37
SCN5A Q14524 2/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
CACNA1C Q13936 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7097450 0.91 KCNH2 (0.39) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL7095963 0.86 KCNH2 (0.40) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL6670398 0.86 KCNH2 (0.37) KCNH2SCN5A
SCHEMBL6370734 0.84 KCNH2 (0.43) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL6669254 0.83
SCHEMBL7097663 0.82 KCNH2 (0.37) KCNH2SCN5A
SCHEMBL6670242 0.82
SCHEMBL6370722 0.81 KCNH2 (0.44) KCNH2SCN5ACYP1A2CYP3A4CYP2D6
SCHEMBL6670217 0.81 CACNA1F (0.33) KCNH2CACNA1C
SCHEMBL7093708 0.80 KCNH2 (0.39) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401830-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2004-03-31 EP claimed
WO-2002102793-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2002-12-27 WO claimed