SCHEMBL6673100

SCHEMBL6673100

CC(CN1c2nc(-c3ccncc3)cc(=O)n2CCC1(C)C)c1ccccc1.CC(CN1c2nc(-c3ccncc3)cc(=O)n2CCC1(C)C)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.43
USP19 O94966 4/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CDC7 O00311 1/20 0.38
ROCK2 O75116 1/20 0.38
MAP4K4 O95819 1/20 0.38
PIM1 P11309 1/20 0.38
PRKACA P17612 1/20 0.38
HIPK2 Q9H2X6 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4871797 1.00 GSK3B (0.43) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL6673105 1.00 GSK3B (0.43) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL4871806 1.00 GSK3B (0.43) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL4872254 1.00 GSK3B (0.43) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL4871119 0.90 GSK3B (0.51) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL4871122 0.90 GSK3B (0.51) GSK3BUSP19CYP1A2CYP2D6CDC7
SCHEMBL4871116 0.90 GSK3B (0.51) GSK3BUSP19CYP1A2CYP2D6CDC7
Hydrochloric Acid SCHEMBL4865765 0.89 GSK3B (0.50) GSK3BUSP19CYP1A2CYP2D6CDC7
Hydrochloric Acid SCHEMBL4865769 0.89 GSK3B (0.50) GSK3BUSP19CYP1A2CYP2D6CDC7
Hydrochloric Acid SCHEMBL4865758 0.89 GSK3B (0.50) GSK3BUSP19CYP1A2CYP2D6CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430057-A2 SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO 1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO 1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES Sanofi-Aventis (FR) 2004-06-23 EP claimed
WO-2003027116-A2 SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES SANOFI-SYNTHELABO (FR) 2003-04-03 WO claimed